Yazar "Tala, Srinivasa R." için listeleme
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Benzotriazole-Mediated Syntheses of Depsipeptides and Oligoesters
Avan, İlker; Tala, Srinivasa R.; Steel, Peter J.; Katritzky, Alan R. (American Chemical Society, 2011)Reactions of O-Pg(alpha-hydroxyacyl)benzotriazoles with (a) unprotected alpha-hydroxycarboxylic acids, (b) amino acids, and (c) amines afforded, respectively, chirally pure (a) oligoesters, (b) depsidipeptides, and (c) ... -
Design, synthesis, and biological activity of a novel series of 2,5-disubstituted furans/pyrroles as HIV-1 fusion inhibitors targeting gp41
Jiang, Shibo; Tala, Srinivasa R.; Lu, Hong; Zou, Peng; Avan, İlker; İbrahim, Tarek S.; Katritzky, Alan R. (Pergamon-Elsevier Science LTD, 2011)Based on molecular docking analysis of earlier results, we designed a series of 2,5-disubstituted furans/pyrroles (5a-h) as HIV-1 entry inhibitors. Compounds were synthesized by Suzuki-Miyaura cross coupling, followed by ... -
Design, Synthesis, and Biological Activity of Novel 5-((Arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones as HIV-1 Fusion Inhibitors Targeting gp41
Jiang, Shibo; Tala, Srinivasa R.; Lu, Hong; Abo-Dya, Nader E.; Avan, İlker; Gyanda, Kapil; Debnath, Asım K. (American Chemical Society, 2011)On the basis of our earlier molecular docking analysis, we designed and synthesized 5-((arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones (12a-o) as HIV-1 entry inhibitors. Compounds ... -
Efficient preparation of aminoxyacyl amides, aminoxy hybrid peptides and a-aminoxy peptides
Tala, Srinivasa R.; Avan, İlker; Katritzky, Alan R. (American Chemical Society, 2010)… -
Efficient Preparation of Aminoxyacyl Amides, Aminoxy Hybrid Peptides, and alpha-Aminoxy Peptides
Katritzky, Alan R.; Avan, İlker; Tala, Srinivasa R. (American Chemical Society, 2009)N-(Pg-alpha-aminoxy acids) 1a-g are converted to N-(Pg-alpha-aminoxyacyl)benzotriazoles 2a-g, Which react under mild conditions with amines, alpha-amino acids/alpha-dipeptides, and alpha-aminoxy acids to give aminoxyacyl ...