Yazar "Jiang, Shibo" için listeleme
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Design, synthesis, and biological activity of a novel series of 2,5-disubstituted furans/pyrroles as HIV-1 fusion inhibitors targeting gp41
Jiang, Shibo; Tala, Srinivasa R.; Lu, Hong; Zou, Peng; Avan, İlker; İbrahim, Tarek S.; Katritzky, Alan R. (Pergamon-Elsevier Science LTD, 2011)Based on molecular docking analysis of earlier results, we designed a series of 2,5-disubstituted furans/pyrroles (5a-h) as HIV-1 entry inhibitors. Compounds were synthesized by Suzuki-Miyaura cross coupling, followed by ... -
Design, Synthesis, and Biological Activity of Novel 5-((Arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones as HIV-1 Fusion Inhibitors Targeting gp41
Jiang, Shibo; Tala, Srinivasa R.; Lu, Hong; Abo-Dya, Nader E.; Avan, İlker; Gyanda, Kapil; Debnath, Asım K. (American Chemical Society, 2011)On the basis of our earlier molecular docking analysis, we designed and synthesized 5-((arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones (12a-o) as HIV-1 entry inhibitors. Compounds ...