Yazar "Karaburun, Ahmet Çağrı" için listeleme
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Bazı 1-[2-(sübstitüe pirol-1-il) etil]-2-metil-5-nitroimidazol türevlerinin sentezi ve antimikrobiyal etkilerinin araştırılması
Karaburun, Ahmet Çağrı (Anadolu Üniversitesi, 1997)Bu çalışmada, 1-[2-(sübstitüe pirol-1-il)etil]-2-metil-5- nitroimidazol türevleri, metronidazol bileşiğinden hazırlanan 2-(2- metil-5-nitro-1H-imidazolil)etilamin dihihroklorür bileşiğinin, beş değişik 1,4-dikarbonil ... -
Bazı 6-[4-(sübstitüe pirol-1-il]-4,5-dihidro-3(2H)-piridazinon ve 1(2H)-ftalazinon türevlerinin sentezi ve antihipertansif etkilerinin araştırılması
Karaburun, Ahmet Çağrı (Anadolu Üniversitesi, 2003)Piridazinon türevlerinin kardiyovasküler sistem üzerinde antihipertansif, pozitif inotropik, platelet agregasyon inhibisyonu ve antiastmatİk etkilerinin olduğu literatür araştırmalan sonunda gözlenmiştir. 6-Aril-3(2H)-piridazinon ... -
New chroman-4-one/thiochroman-4-one derivatives as potential anticancer agents
Demirayak, Şeref; Yurttaş, Leyla; Gündoğdu-Karaburun, Nalan; Karaburun, Ahmet Çağrı; Kayagil, İsmail (Elsevier Science BV, 2017)The synthesis of 3-[3/4-(2-aryl-2-oxoethoxy) arylidene] chroman/thiochroman-4-one derivatives (1-34) and evaluation of their anticancer activities were aimed in this work. Final compounds were obtained in multistep synthesis ... -
Some 1-substituted 3-aryl-1,4-dihydro-1,2,4-triazino[4,3-a]- benzimidazoles and their vasodilatory activities
Demirayak, Şeref; Benkli, Kadriye; Karaburun, Ahmet Çağrı (Societa Chimica Italiana, 1997)In this study, some 1-substituted 3-aryl-1,4-dihydro-1,2,4- triazino[4,3-a]benzimidazole derivatives were synthesized, their structures were elucidated, and their vasodilatory activities were examined. It was found that ... -
Some pyridazinone and phthalazinone derivatives and their vasodilator activities
Demirayak, Şeref; Karaburun, Ahmet Çağrı; Kayagil, İsmail; Erol, K.; Sırmagül, Başar (Pharmaceutical Society of Korea, 2004)In this study, 6-[(4-arylidene-2-phenyl-5-oxoimidazolin-1-yl)phenyl]-4,5- dihydro-3(2H)-pyridazinone and 4-[(4-arylidene-2-phenyl-5-oxoimidazolin-1-yl) phenyl]-1(2H)-phthalazinone derivatives were synthesized by reacting ... -
Some pyrrole substituted aryl pyridazinone and phthalazinone derivatives and their antihypertensive activities
In this work, some 2-nonsubstituted/2-methyl-/2-(2-acetyloxyethyl)-6-[4- (substituted pyrrol-1-yl)phenyl]-4,5-dihydro-3(2H)-pyridazinone, derivatives and 2-nonsubstituted/2-methyl- 4-[4-(substituted pyrrol-1-yl)phenyl]-1(2H)- ... -
Some thiazolylaminopyrrole derivatives and their antimicrobial activity
In this study, some ethyl 1-(4-arylthiazol-2-yl)amino-2-methyl-5-aryl-1H-pyrrole-3-carboxylic acid derivatives were obtained by reacting 1-(2-methyl-3-carbethoxy-5-arylpyrrol-1-yl)thioureas with ?-bromoacetophenone ... -
Synthesis and anti-cancer activity evaluation of new aurone derivatives
Demirayak, Şeref; Yurttaş, Leyla; Gündoğdu-Karaburun, Nalan; Karaburun, Ahmet Çağrı; Kayagil, İsmail (Taylor & Francis LTD, 2015)In this study, we have synthesized 2-[3-or 4-(2-aryl-2-oxoethoxy) arylidene] benzofuran-3-one derivatives (D1-D38) and evaluated their anti-cancer activities. The final compounds were obtained in multistep synthesis reactions ... -
Synthesis and antibacterial activities of some 1-[2-(substituted pyrrol- 1-yl)ethyl]-2-methyl-5-nitroimidazole derivatives
Demirayak, Şeref; Karaburun, Ahmet Çağrı; Kiraz, N. (Elsevier Masson SAS, 1999)In this study, some 1-[2-(substituted pyrrol-1-yl)ethyl]-2-methyl-5- nitroimidazole derivatives were synthesized by reacting 2-(2-methyl-5-nitro- 1H-imidazolyl)ethylamine dihydrochloride, which was prepared using metronidazole, ... -
Synthesis and antibacterial and antifungal evolution of some ethyl 1- aryloxyacetylamino-5-arylpyrrole-3-carboxylic acid derivatives
In this study some ethyl 1-aryloxyacetylamino-2methyl-5-aryl-1H-pyrrole- 3-carboxylic acid derivatives were obtained by reacting some aryloxyacetylhydrazide and 1-aryl-3-carbethoxy-1,4-pentadione derivatives. The antibacterial ... -
Synthesis and Anticancer Activity of Some 1H-inden-1-one Substituted (Heteroaryl)Acetamide Derivatives
Karaburun, Ahmet Çağrı; Gündoğdu-Karaburun, Nalan; Yurttaş, Leyla; Kayagil, İsmail; Demirayak, Şeref (Bentham Science Publ LTD, 2019)Background: The synthesis of 2-[3/4-((6-substituted-1-oxo-2,3-dihydro-1H-inden-2ylidene) methyl)phenoxy]-N-(heteroaryl)acetamide derivatives and the investigation of their anticancer activity were studied. Methods: ... -
Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2-oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives
Gündoğdu-Karaburun, Nalan; Karaburun, Ahmet Çağrı; Demirayak, Şeref; Kayagil, İsmail; Yurttaş, Leyla (Bentham Science Publ LTD, 2014)The synthesis of 2-[3/ 4-(2-substituted phenyl-2-oxoethoxy) benzylidene]-6-substituted-2,3-dihydro-1H-inden-1one derivatives and the investigation of their anticancer activity were studied. 2-(3- or 4-Hydroxybenzylidene) ... -
Synthesis and Anticandidal Activities of Some Aryl (5-Chloro-Benzofuran-2-yl) Ketoximes
Karaburun, Ahmet Çağrı (Bentham Science Publ LTD, 2019)Background: In this study, some aryl (5-chloro-benzofuran-2-yl) ketoximes and their ethers were synthesised to evaluate their antifungal activity against C. albicans, C. glabrata, C. krusei, and C. parapsilosis. Methods: ... -
Synthesis and antifungal activities of some aryl (3-methyl-benzofuran-2-yl) ketoximes
Benkli, Kadriye; Gündoğdu-Karaburun, N; Karaburun, Ahmet Çağrı; Uçucu, Ümit; Demirayak, Şeref; Kiraz, N (Pharmaceutical Society Korea, 2003)In this study, some aryl (3-methyl-benzofuran-2-yl) ketoximes and their. ethers and esters were synthesised. The structure elucidation of the compounds was performed by IR, H-1-NMR, MASS spectroscopy and elemental analyses. ... -
Synthesis and Antifungal Activities of Some Aryl Naphthofuran Ketoximes
Karaburun, Ahmet Çağrı; Gündoğdu-Karaburun, Nalan; Uçucu, Ümit; Demirayak, Şeref (Bentham Science Publ LTD, 2011)In this study, some aryl naphtho[2,1-b] furan-2-yl ketoximes and their ethers and esters were synthesised. The structure elucidation of the compounds was performed by IR, H-1-NMR and MASS spectroscopic data and elemental ... -
Synthesis and antifungal activities of some aryl(benzofuran-2-yl)ketoximes
Demirayak, Şeref; Uçucu, Ümit; Benkli, Kadriye; Gündoğdu-Karaburun, Nalan; Karaburun, Ahmet Çağrı; Akar, D; Kiraz, N (Elsevier Science Sa, 2002)In this study, some aryl(benzofuran-2-yl)ketoximes and their ethers and esters were synthesised. The structure elucidation of the compounds was performed by IR, H-1 NMR and mass spectroscopic data and elemental analyses ... -
Synthesis and Antifungal Potential of Some Novel Benzimidazole-1,3,4-Oxadiazole Compounds
Karaburun, Ahmet Çağrı; Kaya Çavuşoğlu, Betül; Çevik, Ulviye Acar; Osmaniye, Derya; Sağlık, Begüm Nurpelin; Levent, Serkan; Kaplancıklı, Zafer Asım (MDPI, 2019)Discovery of novel anticandidal agents with clarified mechanisms of action, could be a rationalist approach against diverse pathogenic fungal strains due to the rise of resistance to existing drugs. In support to this ... -
Synthesis and Antiproliferative Activity of 2-arylidene 6-(2-aryl-2-oxoethoxy) Benzofuran-3-one Derivatives
Demirayak, Şeref; Yurttaş, Leyla; Karaburun, Ahmet Çağrı; Gündoğdu-Karaburun, Nalan; Kayagil, İsmail (Bentham Science Publ LTD, 2016)The synthesis of 2-arylidene 6-(2-aryl-2-oxoethoxy) benzofuran-3-one derivatives was reported and selected compounds were determined for their anticancer activity evaluation in National Cancer Institute NCI, USA according ... -
Synthesis and biological activity studies of some new benzofuran derivatives
Karaburun, Ahmet Çağrı; Anadolu Üniversitesi, Sağlık Bilimleri Enstitüsü; Dawbaa, Sam Ali Mohammed Mohammed (Anadolu Üniversitesi -Sağlık Bilimleri Enstitüsü, 2021)Benzofuran, endüstride ve ilaç sektöründe yaygın olarak işlev gören kaynaşmış bisiklik bir yapıdır. Benzofuranın ekonomik faydaları ve sentezleme kolaylığı, onu daha sonraki araştırma çalışmaları için bir kullanışlı bir ... -
Synthesis and cytotoxic and analgesic activities of some 1, 5-diaryl-3-ethoxycarbonylpyrrole derivatives
Demirayak, Şeref; Arslan, Rana; Karaburun, Ahmet Çağrı; Kayagil, İsmail; Seller, Zerrin; Uçucu, Ümit (2006)Some 1,5-diaryl-3-ethoxycarbonyl-2-methylpyrrole derivatives were obtained by reacting 1-aryl-3-ethoxycarbonylpent-1,4-diones and a suitable aniline derivative or sulfanilamide under Paal-Knorr pyrrole synthesis conditions. ...
