Yazar "Abo-Dya, Nader E." için listeleme
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Benzotriazole-Mediated Synthesis of Aza-peptides: En Route to an Aza-Leuenkephalin Analogue
Abo-Dya, Nader E.; Biswas, Suvendu; Başak, Akash; Avan, İlker; Alamry, Khalid A.; Katritzky, Alan R. (American Chemical Society, 2013)Novel N-(N-Pg-azadipeptidoyl)benzotriazoles 20a-e couple efficiently with alpha-amino acids 21a-e, dipeptides 22a-c, aminoxyacetic acid 23a, depsidipeptide 23b, and alpha-hydroxy-beta-phenylpropionic acid 27 yielding, ... -
Design, Synthesis, and Biological Activity of Novel 5-((Arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones as HIV-1 Fusion Inhibitors Targeting gp41
Jiang, Shibo; Tala, Srinivasa R.; Lu, Hong; Abo-Dya, Nader E.; Avan, İlker; Gyanda, Kapil; Debnath, Asım K. (American Chemical Society, 2011)On the basis of our earlier molecular docking analysis, we designed and synthesized 5-((arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones (12a-o) as HIV-1 entry inhibitors. Compounds ... -
Photophysics of novel coumarin-labeled depsipeptides in solution: sensing interactions with SDS micelle via TICT model
Biswas, Suvendu; Avan, İlker; Başak, Akash; Abo-Dya, Nader E.; Asiri, Abdullah; Katritzky, Alan R. (Springer Wien, 2013)N-Acylbenzotriazoles enable the synthesis (69-92 % yield) of blue to green fluorescent coumarin-labeled depsidipeptides 8a-f (quantum yields 0.004-0.97) and depsitripeptides 12a-d (quantum yields 0.02-0.96). Detailed ...